Evigrade
Major

Itraconazole × Methadone

Antifungal, triazole×Synthetic opioid, full mu-receptor agonist

Mechanism

Strong CYP3A4 inhibitor. Methadone rises 2-3 fold.

Symptoms

Sedation, respiratory depression, QT prolongation.

Management

Reduce methadone by 25%, ECG monitoring.

Check the full regimen, not just this pair

Opens the checker with these two drugs prefilled. Add the rest of the regimen and recompute additive risks.

Open checker

Sources

All interactions