Evigrade
Major

Clarithromycin × Ciclosporin

Macrolide antibiotic×Immunosuppressants. Calcineurin inhibitors

Mechanism

Clarithromycin inhibits CYP3A4. Cyclosporine rises 2-3 fold – nephrotoxicity.

Symptoms

Rising creatinine, tremor within 5-7 days.

Management

Reduce cyclosporine by 50%, check blood level on day 3. Better – azithromycin.

Check the full regimen, not just this pair

Opens the checker with these two drugs prefilled. Add the rest of the regimen and recompute additive risks.

Open checker

Sources

All interactions