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Alfa-arbutina

Análogo sintético de la arbutina. Inhibe la tirosinasa y reduce la síntesis de melanina sin citotoxicidad directa sobre los melanocitos.

Brightening

Evidence by route

Topical application

C

Weak evidence. In vitro data, open-label studies, or expert consensus.

In vitro studies and small clinical trials confirm depigmenting effect. Large independent RCTs comparing with other agents (azelaic acid, tranexamic acid) are lacking. Stability in formulas at pH above 5 is questionable.

  • Sugimoto K et al. Chem Pharm Bull. 2005;53(9):1056-1059.

Working concentrations

1–3%

Tolerability and safety

Irritation potential

Low

Allergen risk

Low

Pregnancy

Caution

Skin types

Suitable for

NormalDrySensitiveCombinationOily

Frequently asked questions

¿Es seguro Alfa-arbutina durante el embarazo?

Alfa-arbutina se utiliza con precaución durante el embarazo. Conviene consultarlo con un dermatólogo o ginecólogo.

¿Para qué tipos de piel sirve Alfa-arbutina?

Alfa-arbutina es adecuado para: normal, seca, sensible, mixta, grasa.