Evigrade
Major

Rifampicin × Sirolimus

Antituberculous antibiotic×Selective immunosuppressant, mTOR inhibitor

Mechanism

Strong CYP3A4 + P-gp inducer. Sirolimus falls 70% – rejection risk.

Symptoms

Rejection signs.

Management

Alternative TB regimen. If rifampicin necessary – triple sirolimus dose.

Check the full regimen, not just this pair

Opens the checker with these two drugs prefilled. Add the rest of the regimen and recompute additive risks.

Open checker

Sources

All interactions